Structure-Guided Design of IACS-9571, a Selective High-Affinity Dual TRIM24-BRPF1 Bromodomain Inhibitor

Wylie S. Palmer, Guillaume Poncet-Montange, Gang Liu, Alessia Petrocchi, Naphtali Reyna, Govindan Subramanian, Jay Theroff, Anne Yau, Maria Kost-Alimova, Jennifer P. Bardenhagen, Elisabetta Leo, Hannah E. Shepard, Trang N. Tieu, Xi Shi, Yanai Zhan, Shuping Zhao, Michelle C. Barton, Giulio Draetta, Carlo Toniatti, Philip JonesMary Geck Do, Jannik N. Andersen

Research output: Contribution to journalArticlepeer-review

119 Scopus citations

Fingerprint

Dive into the research topics of 'Structure-Guided Design of IACS-9571, a Selective High-Affinity Dual TRIM24-BRPF1 Bromodomain Inhibitor'. Together they form a unique fingerprint.

Medicine & Life Sciences

Chemical Compounds